About 22 results found for searched term "Bradykinin Receptor" (0.127 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M3947 | ELN 441958 | Bradykinin Receptor |
| ELN-441958 is a potent, neutral, competitive and selective oral bioavailable bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. | ||
| M10164 | Icatibant (HOE 140) acetate | Bradykinin Receptor |
| HOE 140 acetate | ||
| Icatibant (HOE-140) acetate is a potent and specific peptide antagonist of bradykinin B2 receptor, with IC50 value of 1.07 nM and Ki value of 0.798 nM, respectively. | ||
| M13916 | Icatibant | Bradykinin Receptor |
| HOE 140 | ||
| Icatibant (HOE-140) is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively. | ||
| M27862 | Fasitibant chloride | Bradykinin Receptor |
| MEN16132 free base | ||
| Fasitibant chloride (MEN16132 free base) is a potent and selective nonpeptide bradykinin B2 receptor (B2R) antagonist. Fasitibant chloride reduces joint pain and diminishes joint oedema in Carrageenan-induced arthritis rat model. | ||
| M30761 | Fasitibant chloride hydrochloride | Bradykinin Receptor |
| MEN16132 | ||
| Fasitibant chloride hydrochloride (MEN16132) is a potent, selective, high affinity, and long-lasting nonpeptide bradykinin B2 (BK2) receptor antagonist. Fasitibant chloride hydrochloride has proinflammatory effects and can be used for the research of osteoarthritis and rheumatoid arthritis. | ||
| M30763 | Fasitibant free base | Bradykinin Receptor |
| Fasitibant (free base) is a potent, selective, high affinity, and long-lasting nonpeptide bradykinin B2 (BK2) receptor antagonist. Fasitibant (free base) has proinflammatory effects and can be used for the research of osteoarthritis and rheumatoid arthritis. | ||
| M41786 | Lys-Bradykinin | Bradykinin Receptor |
| Lys-Bradykinin, a kind of kallidin and bradykinin receptor ligand, can be generated by kininogen protein through enzymatic cleavage by the protease kallikrein. | ||
| M41788 | NPC-567 | Bradykinin Receptor |
| NPC-567 is a bradykinin B2 receptor antagonist. | ||
| M45242 | Deucrictibant | Bradykinin Receptor |
| Deucrictibant is a novel, potent, orally active small molecule bradykinin B2 receptor antagonist. | ||
| M53237 | R715 | Bradykinin Receptor |
| R715 is a selective bradykinin B1 receptor antagonist. | ||
| M53238 | B 9430 | Bradykinin Receptor |
| B 9430 is a potent bradykinin B1/B2 receptor antagonist. | ||
| M53242 | Lys-(Des-Arg9, Leu8)-Bradykinin | Bradykinin Receptor |
| Lys-(Des-Arg9,Leu8)-Bradykinin is a bradykinin B1 receptor antagonist. | ||
| M53243 | Sar-[D-Phe8]-des-Arg9-Bradykinin | Bradykinin Receptor |
| Sar-[D-Phe8]-des-Arg9-Bradykinin is a agonist of B1 receptor. | ||
| M53244 | Des-Arg9-[Leu8]-Bradykinin acetate | Bradykinin Receptor |
| Des-Arg9-[Leu8]-Bradykinin acetate is potent bradykinin receptor 1 (B1R) antagonist. | ||
| M53245 | [Phe8Ψ(CH-NH)Arg9]-Bradykinin | Bradykinin Receptor |
| [Phe8Ψ(CH-NH)Arg9]-Bradykinin is a selective Bradykinin receptor B2 agonist (not cleaved by protein kinase I/II). | ||
| M53246 | [Des-Arg9]-Bradykinin | Bradykinin Receptor |
| [Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors. | ||
| M53248 | Lys-[Des-Arg9]Bradykinin | Bradykinin Receptor |
| Lys-[Des-Arg9]Bradykinin, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. | ||
| M53889 | [Des-Arg9]-Bradykinin acetate | Bradykinin Receptor |
| [Des-Arg9]-Bradykinin acetate is a Bradykinin B1 receptor agonist that displays selectivity for B1 over B2 receptors. | ||
| M54078 | [Tyr8] Bradykinin | Bradykinin Receptor |
| [Tyr8] Bradykinin is a B2 kinin receptor agonist. | ||
| M54123 | Lobradimil | Bradykinin Receptor |
| Lobradimil (RMP 7), a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). | ||
| M54164 | Lys-[Des-Arg9]Bradykinin TFA | Bradykinin Receptor |
| Lys-[Des-Arg9]Bradykinin TFA, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. | ||
| M54281 | [Hyp3]-Bradykinin | Bradykinin Receptor |
| [Hyp3]-Bradykinin, naturally occurring peptide hormone, is a bradykinin receptor agonist. | ||
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